ANILERIDINE%DRUGBANK%DB00913	Anileridine	OPRM1	
INTERFERON ALFA-2A%DRUGBANK%DB00034	Interferon alfa-2a	IFNAR2	IFNAR1	
MONOBENZONE%DRUGBANK%DB00600	Monobenzone	TYR	
PHENACETIN%DRUGBANK%DB03783	Phenacetin	IMPDH1	PTGS1	
TIXOCORTOL%DRUGBANK%DB09091	Tixocortol	HDAC2	NR3C1	
DICHLOROACETIC ACID%DRUGBANK%DB08809	Dichloroacetic acid	GSTZ1	PDK1	
MEPHENTERMINE%DRUGBANK%DB01365	Mephentermine	DRD2	ADRA1A	ADRB1	
IFENPRODIL%DRUGBANK%DB08954	Ifenprodil	KCNJ5	KCNJ6	CELA1	GRIN2B	KCNJ3	GRIN1	
CAPROMAB PENDETIDE%DRUGBANK%DB00089	Capromab pendetide	FOLH1	
METHYPRYLON%DRUGBANK%DB01107	Methyprylon	GABRA1	
ISOFLUROPHATE%DRUGBANK%DB00677	Isoflurophate	BCHE	ACHE	TF	
IBUPROXAM%DRUGBANK%DB08955	Ibuproxam	CXCR1	ALOX5	CXCR2	
TROPISETRON%DRUGBANK%DB11699	Tropisetron	ERBB2	HTR3A	
FLUTICASONE%DRUGBANK%DB13867	Fluticasone	PLA2G4A	PGR	NR3C2	NR3C1	
TELAPREVIR%DRUGBANK%DB05521	Telaprevir	SLCO1B1	SLCO2B1	
EFLORNITHINE%DRUGBANK%DB06243	Eflornithine	ODC1	
DEXKETOPROFEN%DRUGBANK%DB09214	Dexketoprofen	PTGS2	PTGS1	
HALOTHANE%DRUGBANK%DB01159	Halothane	GRIN3A	GNG2	KCNMA1	KCNJ6	RHO	KCNN4	KCNK3	KCNJ3	GABRA1	NPSR1	KCNK9	ATP2B1	MT-ND1	GLRA1	GRIN3B	GRIN2A	
LERCANIDIPINE%DRUGBANK%DB00528	Lercanidipine	CACNA2D1	CACNG1	
THIOPENTAL%DRUGBANK%DB00599	Thiopental	GABRA4	GABRA3	GRIK2	GABRA2	GRIA2	GABRA1	CHRM3	FAAH	GABRA6	GABRA5	CHRNA4	CHRNA7	
CATUMAXOMAB%DRUGBANK%DB06607	Catumaxomab	FCGR3A	FCGR2A	FCGR3B	EPCAM	FCGR1A	CD3E	
SOMATOSTATIN%DRUGBANK%DB09099	Somatostatin	OPRM1	OPRD1	SSTR1	SSTR2	SSTR3	SSTR4	SSTR5	
PIPERACETAZINE%DRUGBANK%DB06808	Piperacetazine	DRD2	
SPARFLOXACIN%DRUGBANK%DB01208	Sparfloxacin	TOP2A	
HYDROCORTISONE CYPIONATE%DRUGBANK%DB14541	Hydrocortisone cypionate	HSD11B2	ANXA1	HSD3B1	NR3C1	
MORICIZINE%DRUGBANK%DB00680	Moricizine	SCN5A	
LEVAMISOLE%DRUGBANK%DB00848	Levamisole	CHRNA3	ALPL	ALPG	
DOPEXAMINE%DRUGBANK%DB12313	Dopexamine	DRD2	
VALDECOXIB%DRUGBANK%DB00580	Valdecoxib	CA3	CA2	PTGS2	
VIDARABINE%DRUGBANK%DB00194	Vidarabine	ADORA2B	
INTERFERON ALFA%DRUGBANK%DB05258	Interferon alfa	IFNAR1	
DIENESTROL%DRUGBANK%DB00890	Dienestrol	SHBG	ESR1	
SODIUM CARBONATE%DRUGBANK%DB09460	Sodium carbonate	CA2	CA1	CA4	CA9	
ETHINAMATE%DRUGBANK%DB01031	Ethinamate	CA2	CA1	
DIPHENIDOL%DRUGBANK%DB01231	Diphenidol	CHRM1	CHRM4	CHRM3	CHRM2	
PEGAPTANIB%DRUGBANK%DB04895	Pegaptanib	NRP1	VEGFA	
DIPIVEFRIN%DRUGBANK%DB00449	Dipivefrin	ADRA1A	ADRB2	ADRA2A	BCHE	ACHE	ADRB1	
APROTININ%DRUGBANK%DB06692	Aprotinin	PRSS1	KLK1	CTRB1	PLG	
ESTRAMUSTINE%DRUGBANK%DB01196	Estramustine	MAP2	MAP1A	ESR1	ESR2	
TRILOSTANE%DRUGBANK%DB01108	Trilostane	HSD3B1	ESR1	ESR2	HSD3B2	
TEGASEROD%DRUGBANK%DB01079	Tegaserod	HTR2A	HTR4	HTR2B	HTR2C	
AUROTHIOGLUCOSE%DRUGBANK%DB09121	Aurothioglucose	ADCY2	ADCY1	ADCY5	
ABARELIX%DRUGBANK%DB00106	Abarelix	GNRHR	
MEPENZOLATE%DRUGBANK%DB04843	Mepenzolate	CHRM1	CHRM5	CHRM3	
NIALAMIDE%DRUGBANK%DB04820	Nialamide	MAOB	MAOA	COMT	
LASOFOXIFENE%DRUGBANK%DB06202	Lasofoxifene	CNR2	ESR1	ESR2	
PHENPROCOUMON%DRUGBANK%DB00946	Phenprocoumon	VKORC1	
AMINOHIPPURIC ACID%DRUGBANK%DB00345	Aminohippuric acid	SLC22A8	
PAPAIN%DRUGBANK%DB11193	Papain	TLR4	
D-SERINE%DRUGBANK%DB03929	D-Serine	GRIN1	GLRA1	SERPINB3	
GEMEPROST%DRUGBANK%DB08964	Gemeprost	PTGER3	PTGER2	
CAPRYLIC ACID%DRUGBANK%DB04519	Caprylic acid	PPARA	
MESORIDAZINE%DRUGBANK%DB00933	Mesoridazine	HTR2A	DRD2	
HEXACHLOROPHENE%DRUGBANK%DB00756	Hexachlorophene	GLUD1	SDHD	ESR1	
LUMIRACOXIB%DRUGBANK%DB01283	Lumiracoxib	PTGS2	PTGS1	
IOPODIC ACID%DRUGBANK%DB09333	Iopodic acid	DIO3	
INGENOL MEBUTATE%DRUGBANK%DB05013	Ingenol mebutate	PRKCD	PRKCA	
BUTABARBITAL%DRUGBANK%DB00237	Butabarbital	GRIK2	GRIA1	GRIK5	GRIA2	GABRA1	GRIK3	CHRNA10	GRIK4	GRIK1	GRIA3	GRIA4	
LITHIUM CATION%DRUGBANK%DB01356	Lithium cation	IMPA1	IMPA2	GRIA3	GSK3B	
NEUROPEPTIDE Y%DRUGBANK%DB11788	Neuropeptide Y	NPY2R	NPY1R	
NYLIDRIN%DRUGBANK%DB06152	Nylidrin	CACNA1I	IFNAR2	
PROBUCOL%DRUGBANK%DB01599	Probucol	ABCA1	CES1	
ALBIGLUTIDE%DRUGBANK%DB09043	Albiglutide	GLP1R	
FOSPROPOFOL%DRUGBANK%DB06716	Fospropofol	GABRB3	GABRB2	
BROMFENAC%DRUGBANK%DB00963	Bromfenac	PTGS2	PTGS1	
ETRETINATE%DRUGBANK%DB00926	Etretinate	RXRB	RARG	RXRA	RARA	RARB	RXRG	
5-O-PHOSPHONO-ALPHA-D-RIBOFURANOSYL DIPHOSPHATE%DRUGBANK%DB01632	5-O-phosphono-alpha-D-ribofuranosyl diphosphate	HPRT1	UCKL1	APRT	
LEPIRUDIN%DRUGBANK%DB00001	Lepirudin	F2	
DROTAVERINE%DRUGBANK%DB06751	Drotaverine	PDE4A	CACNA1C	
ROXITHROMYCIN%DRUGBANK%DB00778	Roxithromycin	ABCB1	
TAUROURSODEOXYCHOLIC ACID%DRUGBANK%DB08834	Tauroursodeoxycholic acid	ITGA5	
ABCIXIMAB%DRUGBANK%DB00054	Abciximab	FCGR2A	VTN	ITGB3	ITGA2B	FCGR2B	
FLECAINIDE%DRUGBANK%DB01195	Flecainide	SCN5A	KCNH2	RYR2	SCN4A	
OMACETAXINE MEPESUCCINATE%DRUGBANK%DB04865	Omacetaxine mepesuccinate	RPL3	
SULPIRIDE%DRUGBANK%DB00391	Sulpiride	DRD2	DRD3	DRD4	CA3	CA2	
BEMIPARIN%DRUGBANK%DB09258	Bemiparin	SERPIND1	F10	SERPINC1	
UROFOLLITROPIN%DRUGBANK%DB00094	Urofollitropin	FSHR	
ONDANSETRON%DRUGBANK%DB00904	Ondansetron	HTR3A	HTR4	OPRM1	HTR1A	HTR1B	
PHENYLPROPANOLAMINE%DRUGBANK%DB00397	Phenylpropanolamine	ADRB2	ADRA2A	TERT	DRD1	ADRB1	
DYPHYLLINE%DRUGBANK%DB00651	Dyphylline	PDE4A	NT5E	ADORA2A	PDE4D	PDE4C	PDE4B	ADORA1	
STREPTOKINASE%DRUGBANK%DB00086	Streptokinase	F2R	PLG	
INDORAMIN%DRUGBANK%DB08950	Indoramin	ADRA1D	ADRA1A	ADRA2C	ADRA2B	
LYME DISEASE VACCINE (RECOMBINANT OSPA)%DRUGBANK%DB00045	Lyme disease vaccine (recombinant OspA)	TLR2	
PROMAZINE%DRUGBANK%DB00420	Promazine	CHRM1	HTR2A	DRD2	ADRA1A	HRH1	CHRM5	HTR2C	
EZOGABINE%DRUGBANK%DB04953	Ezogabine	KCNQ2	KCNQ3	KCNQ4	KCNQ5	
FENOTEROL%DRUGBANK%DB01288	Fenoterol	ADRB2	ADRB3	ADRB1	
OPRELVEKIN%DRUGBANK%DB00038	Oprelvekin	IL11RA	
HISTRELIN%DRUGBANK%DB06788	Histrelin	GNRHR	
SULFADOXINE%DRUGBANK%DB01299	Sulfadoxine	MAOB	
FORMESTANE%DRUGBANK%DB08905	Formestane	CYP19A1	
NOVOBIOCIN%DRUGBANK%DB01051	Novobiocin	TOP2B	TOP2A	
OXETHAZAINE%DRUGBANK%DB12532	Oxethazaine	GAST	
PEGADEMASE%DRUGBANK%DB00061	Pegademase	GRB2	
PARACHLOROPHENOL%DRUGBANK%DB13154	Parachlorophenol	SCN4A	
ASPARAGINE%DRUGBANK%DB00174	Asparagine	SLC38A1	NARS1	NARS2	ASNS	SLC1A5	ASRGL1	
CALCIUM CARBIMIDE%DRUGBANK%DB09116	Calcium carbimide	ALDH3B2	ALDH2	ALDH1B1	ALDH1A1	
RIBOSTAMYCIN%DRUGBANK%DB03615	Ribostamycin	P4HB	
REMOXIPRIDE%DRUGBANK%DB00409	Remoxipride	HTR2A	DRD2	DRD3	DRD4	SIGMAR1	
ENOXIMONE%DRUGBANK%DB04880	Enoximone	PDE3A	
CYSTINE%DRUGBANK%DB00138	Cystine	CTNS	SLC7A11	
AZATADINE%DRUGBANK%DB00719	Azatadine	HRH1	
PENBUTOLOL%DRUGBANK%DB01359	Penbutolol	ADRB2	HTR1A	HTR1B	ADRB1	
URIDINE%DRUGBANK%DB02745	Uridine	TYMP	LSM6	
RANITIDINE%DRUGBANK%DB00863	Ranitidine	HRH2	ACHE	
ETHYLESTRENOL%DRUGBANK%DB01493	Ethylestrenol	AR	
LEVACETYLMETHADOL%DRUGBANK%DB01227	Levacetylmethadol	CHRNB4	CHRNA3	OPRM1	
NESIRITIDE%DRUGBANK%DB04899	Nesiritide	NPR1	NPR2	NPR3	
RIMONABANT%DRUGBANK%DB06155	Rimonabant	CNR1	GPR55	
TACRINE%DRUGBANK%DB00382	Tacrine	CES1	BCHE	ACHE	
THIORIDAZINE%DRUGBANK%DB00679	Thioridazine	HTR2A	DRD2	ADRA1A	DRD1	ADRA1B	KCNH2	
RAPACURONIUM%DRUGBANK%DB04834	Rapacuronium	CHRM2	
BUTRIPTYLINE%DRUGBANK%DB09016	Butriptyline	HTR2A	HRH1	SLC6A4	
ETHIONAMIDE%DRUGBANK%DB00609	Ethionamide	NFE2L2	
ENPROFYLLINE%DRUGBANK%DB00824	Enprofylline	PDE4A	ADORA2B	NT5E	ADORA2A	ADORA3	PDE4B	ADORA1	
ARZOXIFENE%DRUGBANK%DB06249	Arzoxifene	ESR1	ESR2	
THIETHYLPERAZINE%DRUGBANK%DB00372	Thiethylperazine	DRD2	
TROGLITAZONE%DRUGBANK%DB00197	Troglitazone	ACSL4	PPARG	PPARA	ESRRG	SLC29A1	PPARD	ESRRA	GSTP1	SERPINE1	
IODIPAMIDE%DRUGBANK%DB04711	Iodipamide	ALB	
SERMORELIN%DRUGBANK%DB00010	Sermorelin	GHRHR	
MEBEVERINE%DRUGBANK%DB12554	Mebeverine	CHRM5	
NITRENDIPINE%DRUGBANK%DB01054	Nitrendipine	KCNMA1	CACNA1C	CACNA2D1	CACNB2	CACNA2D2	CACNA1D	CACNA1S	CACNA1H	
DOTATATE GALLIUM GA-68%DRUGBANK%DB13925	Dotatate gallium Ga-68	SSTR2	
PHENOLPHTHALEIN%DRUGBANK%DB04824	Phenolphthalein	SHBG	ESR1	NR1I3	NR1I2	UGT1A9	
ALPHA-LINOLENIC ACID%DRUGBANK%DB00132	alpha-Linolenic acid	PPARG	PPARD	RXRA	ELOVL5	ELOVL2	NR1H4	PPARA	TRPV1	SLC8A1	FADS2	FFAR1	FADS1	PTGS2	
ARACHIDONIC ACID%DRUGBANK%DB04557	Arachidonic Acid	NR1H4	PPARA	PTGS1	RXRA	
BENZOIN%DRUGBANK%DB14020	Benzoin	CES1	
CHLORPROTHIXENE%DRUGBANK%DB01239	Chlorprothixene	CHRM1	HTR2A	DRD2	DRD3	CHRM4	HRH1	CHRM5	HTR1A	DRD1	CHRM3	CHRM2	
DIHYDROTACHYSTEROL%DRUGBANK%DB01070	Dihydrotachysterol	VDR	
METAMFETAMINE%DRUGBANK%DB01577	Metamfetamine	DRD2	MAOB	MAOA	ADRA2C	ADRA2B	ADRA2A	TAAR1	ADRA1B	SLC6A2	SLC6A3	SLC6A4	SLC18A1	SLC18A2	
MOXONIDINE%DRUGBANK%DB09242	Moxonidine	ADRA2C	ADRA2B	ADRA2A	NISCH	
PRENYLAMINE%DRUGBANK%DB04825	Prenylamine	MYLK2	CALM1	
POTASSIUM PERCHLORATE%DRUGBANK%DB09418	Potassium perchlorate	SLC5A5	
PIXANTRONE%DRUGBANK%DB06193	Pixantrone	TOP2B	TOP2A	
ALVERINE%DRUGBANK%DB01616	Alverine	HTR1A	
DACLIZUMAB%DRUGBANK%DB00111	Daclizumab	C1QB	C1QA	FCGR3A	C1R	FCGR2A	IL2RA	FCGR3B	IL2RB	FCGR2C	FCGR1A	C1QC	FCGR2B	
DIGITOXIN%DRUGBANK%DB01396	Digitoxin	ATP1A3	ATP1B3	ATP1A2	ATP1A1	ATP1B2	ATP1B1	
LESINURAD%DRUGBANK%DB11560	Lesinurad	SLC22A12	SLC22A11	
MANIDIPINE%DRUGBANK%DB09238	Manidipine	CACNA1G	CACNA1I	CACNA1C	CACNA1D	CACNA1H	
PIPRADROL%DRUGBANK%DB11584	Pipradrol	DRD1	
CAMPHOR%DRUGBANK%DB01744	Camphor	TRPA1	TRPV3	TRPV1	TRPM8	
CLIOQUINOL%DRUGBANK%DB04815	Clioquinol	OPRK1	
ETORICOXIB%DRUGBANK%DB01628	Etoricoxib	PTGS2	
CHLOROXINE%DRUGBANK%DB01243	Chloroxine	OPRK1	
BROMOCRIPTINE%DRUGBANK%DB01200	Bromocriptine	HTR2A	DRD2	DRD3	ADRA1A	DRD4	HTR1A	HTR1B	DRD1	ADRA1D	ADRA2C	ADRA2B	HTR1D	ADRA2A	HTR7	DRD5	ADRA1B	HTR2B	HTR2C	
ISOFLAVONE%DRUGBANK%DB12007	Isoflavone	PPARG	PPARA	
ADENOSINE PHOSPHATE%DRUGBANK%DB00131	Adenosine phosphate	FBP1	ADCY1	HINT1	PRKAA1	CREB1	ACSS2	ACSL1	PDE4D	ADK	PDE4B	PYGL	PRKAB1	
ARDEPARIN%DRUGBANK%DB00407	Ardeparin	SERPIND1	SERPINC1	
TESTOSTERONE PROPIONATE%DRUGBANK%DB01420	Testosterone propionate	AR	
CHLORPHENOXAMINE%DRUGBANK%DB09007	Chlorphenoxamine	HRH1	
BUTAMBEN%DRUGBANK%DB11148	Butamben	TRPA1	TRPV4	KCNJ1	CACNG1	
NOMIFENSINE%DRUGBANK%DB04821	Nomifensine	DRD2	MPO	MAOB	MAOA	SLC6A2	SLC6A3	SLC6A4	SLC18A2	
ESTRADIOL BENZOATE%DRUGBANK%DB13953	Estradiol benzoate	ESRRG	MT-ATP6	NCOA2	BECN1	GPER1	HSD17B2	ESR1	ESR2	NR1I2	CHRNA4	
METHOXYFLURANE%DRUGBANK%DB01028	Methoxyflurane	GRIA1	GABRA1	KCNA1	ATP2C1	MT-ND1	GLRA1	
CARBOXIN%DRUGBANK%DB04657	Carboxin	SDHA	
SULODEXIDE%DRUGBANK%DB06271	Sulodexide	SERPIND1	SERPINC1	
ENFLURANE%DRUGBANK%DB00228	Enflurane	CACNG1	GRIN1	GABRA1	ATP2C1	ATP2A1	GLRA1	
CLOFIBRATE%DRUGBANK%DB00636	Clofibrate	PPARA	LPL	
DINOPROST%DRUGBANK%DB12789	Dinoprost	PTGDR2	PTGER3	PTGER1	TBXA2R	PTGDR	PTGER4	PTGFR	PTGER2	
AMINOPTERIN%DRUGBANK%DB08878	Aminopterin	PDF	
AZACYCLONOL%DRUGBANK%DB19381	AZACYCLONOL	HRH1	
MEPHENYTOIN%DRUGBANK%DB00532	Mephenytoin	SCN5A	NR1I2	
GUANETHIDINE%DRUGBANK%DB01170	Guanethidine	SLC6A2	
DIETHYLSTILBESTROL%DRUGBANK%DB00255	Diethylstilbestrol	AR	ESRRG	NCOA2	ESRRB	SHBG	ESR1	ESR2	ESRRA	NR1I2	
HALOFANTRINE%DRUGBANK%DB01218	Halofantrine	CALM3	CALM2	KCNH2	CALM1	
YOHIMBINE%DRUGBANK%DB01392	Yohimbine	HTR2A	DRD2	DRD3	ADRA2C	KCNJ1	ADRA2B	HTR1D	ADRA2A	HTR1A	HTR1B	HTR2B	HTR2C	
AMRINONE%DRUGBANK%DB01427	Amrinone	PDE4A	PDE3B	TNF	PDE3A	
TUBOCURARINE%DRUGBANK%DB01199	Tubocurarine	HTR3A	CHRNA2	ACHE	CHRNA7	
HYDROFLUMETHIAZIDE%DRUGBANK%DB00774	Hydroflumethiazide	KCNMA1	CA2	CA12	ATP1A1	CA1	SLC12A1	CA4	CA7	CA9	
DEXIBUPROFEN%DRUGBANK%DB09213	Dexibuprofen	SLC15A1	BCL2	PPARG	PPARA	PLAT	GP1BA	CFTR	S100A7	PTGS2	PTGS1	THBD	FABP2	
ALOSETRON%DRUGBANK%DB00969	Alosetron	HTR3A	HTR3B	
EFALIZUMAB%DRUGBANK%DB00095	Efalizumab	ITGAX	ITGAL	
BENTIROMIDE%DRUGBANK%DB00522	Bentiromide	HPN	
PERAZINE%DRUGBANK%DB12710	Perazine	DRD2	
IPRONIAZID%DRUGBANK%DB04818	Iproniazid	MAOB	MAOA	
TOCAINIDE%DRUGBANK%DB01056	Tocainide	SCN5A	
LEVOSIMENDAN%DRUGBANK%DB00922	Levosimendan	KCNJ8	KCNJ11	TNNC1	PDE3A	
EDOXUDINE%DRUGBANK%DB13421	Edoxudine	TK1	
ETOPERIDONE%DRUGBANK%DB09194	Etoperidone	CHRM1	HTR2A	DRD2	ADRA1A	ADRA2A	HTR2C	
BENZBROMARONE%DRUGBANK%DB12319	Benzbromarone	ABCC1	CYP2C19	SLC22A12	CYP2C9	ANO1	
DYDROGESTERONE%DRUGBANK%DB00378	Dydrogesterone	PGR	
MUROMONAB%DRUGBANK%DB00075	Muromonab	CD3G	CD247	CD3D	FCGR3B	CD3E	
METOCURINE IODIDE%DRUGBANK%DB00416	Metocurine iodide	CHRNB2	CHRNA2	CHRNA4	
SIBUTRAMINE%DRUGBANK%DB01105	Sibutramine	SLC6A2	SLC6A3	SLC6A4	
PROPANOIC ACID%DRUGBANK%DB03766	Propanoic acid	GPHN	
PHENYLBUTAZONE%DRUGBANK%DB00812	Phenylbutazone	PTGIS	PTGS2	PTGS1	
CARPHENAZINE%DRUGBANK%DB01038	Carphenazine	DRD2	DRD5	DRD1	
INOSITOL%DRUGBANK%DB13178	Inositol	APP	
DANAPAROID%DRUGBANK%DB06754	Danaparoid	SERPINC1	
OXPRENOLOL%DRUGBANK%DB01580	Oxprenolol	ADRB2	ADRB3	ADRB1	
FLUBENDAZOLE%DRUGBANK%DB08974	Flubendazole	TUBA1A	
ANISTREPLASE%DRUGBANK%DB00029	Anistreplase	PLG	FGA	SERPINE1	
TERFENADINE%DRUGBANK%DB00342	Terfenadine	CHRM1	CHRM4	HRH1	CHRM5	CHRM3	KCNH2	CHRM2	
PROCATEROL%DRUGBANK%DB01366	Procaterol	ADRB2	
UROKINASE%DRUGBANK%DB00013	Urokinase	NID1	SERPINA5	PLG	ST14	SERPINB2	PLAU	PLAUR	SERPINE1	LRP2	
CISAPRIDE%DRUGBANK%DB00604	Cisapride	HTR2A	HTR3A	HTR4	KCNH2	
BITOLTEROL%DRUGBANK%DB00901	Bitolterol	ADRB2	ADRB3	
KETAZOLAM%DRUGBANK%DB01587	Ketazolam	GABRA1	
PREGNENOLONE%DRUGBANK%DB02789	Pregnenolone	SULT2B1	ESRRA	NR1I2	
DEXTROPROPOXYPHENE%DRUGBANK%DB00647	Dextropropoxyphene	OPRK1	OPRM1	GRIN1	OPRD1	
CHOLECYSTOKININ%DRUGBANK%DB08862	Cholecystokinin	CCKAR	CCKBR	PRKCB	EGF	RAF1	MAPK3	
HUPERZINE A%DRUGBANK%DB04864	Huperzine A	AMY2A	ACHE	ALOX5	
UMBRALISIB%DRUGBANK%DB14989	Umbralisib	ABL1	PIK3CD	CSNK1E	
METHYSERGIDE%DRUGBANK%DB00247	Methysergide	HTR2A	HTR7	HTR1A	HTR1B	HTR1E	HTR1F	HTR2B	HTR2C	
CHLORPHENTERMINE%DRUGBANK%DB01556	Chlorphentermine	SLC6A4	
BENDAZAC%DRUGBANK%DB13501	Bendazac	PTGS2	PTGS1	
MAFENIDE%DRUGBANK%DB06795	Mafenide	CA14	CA2	CA12	CA4	CA6	
ENCAINIDE%DRUGBANK%DB01228	Encainide	SCN5A	
CERIVASTATIN%DRUGBANK%DB00439	Cerivastatin	HMGCR	
QUINAGOLIDE%DRUGBANK%DB09097	Quinagolide	DRD2	DRD1	
TOSITUMOMAB%DRUGBANK%DB00081	Tositumomab	MS4A1	FCGR2B	
METAMIZOLE%DRUGBANK%DB04817	Metamizole	PTGS1	
DEXTROTHYROXINE%DRUGBANK%DB00509	Dextrothyroxine	TPO	THRB	THRA	
ALUMINIUM%DRUGBANK%DB01370	Aluminium	KLK1	APP	ATP1A1	TF	
AVEXITIDE%DRUGBANK%DB14806	Avexitide	GLP1R	
DIMETACRINE%DRUGBANK%DB08996	Dimetacrine	ACHE	
INTERFERON ALFACON-1%DRUGBANK%DB00069	Interferon alfacon-1	IFNAR2	IFNAR1	
GUANABENZ%DRUGBANK%DB00629	Guanabenz	ADRA2B	ADRA2A	
CLOFEDANOL%DRUGBANK%DB04837	Clofedanol	HRH1	
DIFLUOCORTOLONE%DRUGBANK%DB09095	Difluocortolone	ANXA3	NR3C1	
DIETHYLCARBAMAZINE%DRUGBANK%DB00711	Diethylcarbamazine	PTGS1	ALOX5	
PIRENZEPINE%DRUGBANK%DB00670	Pirenzepine	CHRM1	
ALEFACEPT%DRUGBANK%DB00092	Alefacept	FCGR3A	FCGR3B	CD2	CD58	
PIPECURONIUM%DRUGBANK%DB01338	Pipecuronium	CHRM3	CHRNA2	CHRM2	
BELANTAMAB MAFODOTIN%DRUGBANK%DB15719	Belantamab mafodotin	TNFRSF17	
AMSACRINE%DRUGBANK%DB00276	Amsacrine	ALB	ORM1	KCNH2	TOP2B	TOP2A	
CHYMOPAPAIN%DRUGBANK%DB06752	Chymopapain	PRG2	
PEGINESATIDE%DRUGBANK%DB08894	Peginesatide	EPOR	
AMYLOCAINE%DRUGBANK%DB09088	Amylocaine	SCN1A	
DEXFENFLURAMINE%DRUGBANK%DB01191	Dexfenfluramine	SLC6A4	HTR2C	
PIRBUTEROL%DRUGBANK%DB01291	Pirbuterol	ADRB2	ADRB1	
PERGOLIDE%DRUGBANK%DB01186	Pergolide	HTR2A	DRD2	DRD3	ADRA1A	DRD4	HTR1A	HTR1B	DRD1	ADRA1D	HTR1D	ADRA2A	DRD5	ADRA1B	HTR2B	HTR2C	
RILMENIDINE%DRUGBANK%DB11738	Rilmenidine	ADRA2C	ADRA2A	
CHLORMERODRIN%DRUGBANK%DB00534	Chlormerodrin	SLC12A1	ALDH5A1	
AMINEPTINE%DRUGBANK%DB04836	Amineptine	SLC6A2	SLC6A3	SLC6A4	
DEXRAZOXANE%DRUGBANK%DB00380	Dexrazoxane	TOP2B	TOP2A	
AMBENONIUM%DRUGBANK%DB01122	Ambenonium	ACHE	
BUFEXAMAC%DRUGBANK%DB13346	Bufexamac	HDAC6	PTGS2	PTGS1	HDAC10	
MOBOCERTINIB%DRUGBANK%DB16390	Mobocertinib	EGFR	
MIBEFRADIL%DRUGBANK%DB01388	Mibefradil	CACNA1G	CACNB1	CACNB3	CACNA1I	CACNB4	CACNA1C	CACNA1F	CACNB2	CACNA1D	CACNA1S	CACNA1H	
NEFAZODONE%DRUGBANK%DB01149	Nefazodone	HTR2A	ADRA1A	ADRA2A	HTR1A	ADRA1B	SLC6A2	SLC6A3	SLC6A4	KCNH2	HTR2C	
FENFLURAMINE%DRUGBANK%DB00574	Fenfluramine	HTR2A	HTR1D	HTR1A	SLC6A4	SIGMAR1	HTR2B	HTR2C	
SITAXENTAN%DRUGBANK%DB06268	Sitaxentan	EDNRA	EDNRB	
BERBERINE%DRUGBANK%DB04115	Berberine	TERT	BIRC5	
LEVOPROPOXYPHENE%DRUGBANK%DB06793	Levopropoxyphene	OPRM1	
INOSITOL NICOTINATE%DRUGBANK%DB08949	Inositol nicotinate	HCAR2	HCAR3	
DIOXYBENZONE%DRUGBANK%DB11221	Dioxybenzone	SHBG	
LAROPIPRANT%DRUGBANK%DB11629	Laropiprant	PTGDR2	HMGCR	TBXA2R	PTGDR	PTGIR	PTGFR	PTGER2	
TETRACYCLINE%DRUGBANK%DB00759	Tetracycline	PRNP	
ZOXAZOLAMINE%DRUGBANK%DB19372	Zoxazolamine	KCNN2	
DINOPROST TROMETHAMINE%DRUGBANK%DB01160	Dinoprost tromethamine	PTGIR	PTGFR	
HALCINONIDE%DRUGBANK%DB06786	Halcinonide	ESRRG	ESRRB	ESRRA	SMO	
PIPERAZINE%DRUGBANK%DB00592	Piperazine	GABRB3	
FLUPENTIXOL%DRUGBANK%DB00875	Flupentixol	CHRM1	HTR2A	DRD2	DRD3	ADRA1A	DRD4	DRD1	HTR2C	
CHLORAMPHENICOL%DRUGBANK%DB00446	Chloramphenicol	CD55	
DIACEREIN%DRUGBANK%DB11994	Diacerein	CYP2D6	NR1H2	IL1B	CYP1A2	NR1H3	CYP2E1	CYP3A4	CYP2C9	ALOX5	
SUPROFEN%DRUGBANK%DB00870	Suprofen	PTGS2	PTGS1	
ZOTEPINE%DRUGBANK%DB09225	Zotepine	HTR2A	DRD2	HTR7	HTR6	DRD1	SLC6A2	SLC6A4	
METIPRANOLOL%DRUGBANK%DB01214	Metipranolol	ADRB2	ADRB1	
HALAZEPAM%DRUGBANK%DB00801	Halazepam	TSPO	GABRA1	
CLOFAZIMINE%DRUGBANK%DB00845	Clofazimine	PPARG	KCNA3	
BITHIONOL%DRUGBANK%DB04813	Bithionol	CAPN2	ESR1	MCL1	ESR2	
EBASTINE%DRUGBANK%DB11742	Ebastine	HRH1	
NALMEFENE%DRUGBANK%DB06230	Nalmefene	OPRK1	OPRM1	OPRD1	
FERRIC CATION%DRUGBANK%DB13949	Ferric cation	TFRC	
MOLSIDOMINE%DRUGBANK%DB09282	Molsidomine	GUCY1A2	
TOLRESTAT%DRUGBANK%DB02383	Tolrestat	AKR1B1	SIGMAR1	AKR1B10	AKR1A1	
INTERFERON ALFA-N1%DRUGBANK%DB00011	Interferon alfa-n1	IFNAR2	IFNAR1	
KEYHOLE LIMPET HEMOCYANIN%DRUGBANK%DB05299	Keyhole limpet hemocyanin	IL2	
TILARGININE%DRUGBANK%DB11815	Tilarginine	NOS3	
CYCLANDELATE%DRUGBANK%DB04838	Cyclandelate	CACNA2D1	CES1	
CIPROFIBRATE%DRUGBANK%DB09064	Ciprofibrate	PPARA	
FLUSPIRILENE%DRUGBANK%DB04842	Fluspirilene	HTR2A	DRD2	CACNG1	
BIOALLETHRIN%DRUGBANK%DB13746	Bioallethrin	CACNA1G	CACNA1A	CACNA1C	CACNG1	SCN1A	
BEPRIDIL%DRUGBANK%DB01244	Bepridil	CACNA1A	PDE1B	KCNQ1	PDE1A	CACNA2D2	ATP1A1	CACNA1H	KCNH2	TNNC1	CALM1	
ATALUREN%DRUGBANK%DB05016	Ataluren	DMD	
TOLCAPONE%DRUGBANK%DB00323	Tolcapone	COMT	
ACETOHEXAMIDE%DRUGBANK%DB00414	Acetohexamide	KCNJ1	ABCC8	
PHENFORMIN%DRUGBANK%DB00914	Phenformin	PRKAA1	PRKAG1	KCNJ8	PRKAB1	
MIANSERIN%DRUGBANK%DB06148	Mianserin	HTR2A	DRD2	DRD3	ADRA1A	HTR1A	DRD1	HRH4	HTR1F	ADRA2C	ADRA2B	OPRK1	ADRA2A	HRH1	HTR7	HTR6	SLC6A2	SLC6A3	SLC6A4	HTR2B	HTR2C	
1,2-BENZODIAZEPINE%DRUGBANK%DB12537	1,2-Benzodiazepine	TSPO	GABRA1	
BENACTYZINE%DRUGBANK%DB09023	Benactyzine	CHRM5	
MEDROGESTONE%DRUGBANK%DB09124	Medrogestone	PGR	
BROTIZOLAM%DRUGBANK%DB09017	Brotizolam	GABRA1	
LACTOSE%DRUGBANK%DB04465	Lactose	GLTP	LGALS3	GLB1	GLT6D1	
NICORANDIL%DRUGBANK%DB09220	Nicorandil	ABCC9	
MESTRANOL%DRUGBANK%DB01357	Mestranol	ESR1	
BENZQUINAMIDE%DRUGBANK%DB00767	Benzquinamide	CHRM1	CHRM4	HRH1	CHRM5	CHRM3	CHRM2	
DOMATINOSTAT%DRUGBANK%DB17521	Domatinostat	HDAC1	
OXYPHENBUTAZONE%DRUGBANK%DB03585	Oxyphenbutazone	PLA2G2E	ALB	
LENOGRASTIM%DRUGBANK%DB13144	Lenograstim	CSF3R	
ETHOXZOLAMIDE%DRUGBANK%DB00311	Ethoxzolamide	CA3	CA2	CA1	CA4	CA7	
CLOBETASOL%DRUGBANK%DB11750	Clobetasol	PLA2G1B	
METHARBITAL%DRUGBANK%DB00463	Metharbital	GABRA4	GABRA3	GRIK2	GABRG3	GABRA2	GRIA2	GABRA1	GABRA6	GABRA5	CHRNA4	CHRNA7	
MAGNESIUM ACETATE TETRAHYDRATE%DRUGBANK%DB09409	Magnesium acetate tetrahydrate	GRIN1	
ISOPROPAMIDE%DRUGBANK%DB01625	Isopropamide	CHRM4	CHRM3	
GALLAMINE TRIETHIODIDE%DRUGBANK%DB00483	Gallamine triethiodide	CHRM1	CHRM5	CHRNA2	ACHE	CHRM2	
CARPROFEN%DRUGBANK%DB00821	Carprofen	PTGS2	PTGS1	
SOMATREM%DRUGBANK%DB09098	Somatrem	GHR	IGF1R	
OCRIPLASMIN%DRUGBANK%DB08888	Ocriplasmin	SERPINF2	FN1	A2M	
VINDESINE%DRUGBANK%DB00309	Vindesine	TUBB1	
TRIDIHEXETHYL%DRUGBANK%DB00505	Tridihexethyl	CHRM1	CHRM5	CHRM3	CHRM2	
ZILEUTON%DRUGBANK%DB00744	Zileuton	ALOX5	
TRIFLUSAL%DRUGBANK%DB08814	Triflusal	PTGS1	PDE10A	NOS2	NFKB1	
CELIPROLOL%DRUGBANK%DB04846	Celiprolol	ADRA2C	ADRA2B	ADRB2	ADRA2A	ADRB3	ADRB1	
AMLEXANOX%DRUGBANK%DB01025	Amlexanox	S100A13	S100A12	FGF1	IL3	HSP90AA1	
TESTOLACTONE%DRUGBANK%DB00894	Testolactone	CYP19A1	
LOTEPREDNOL%DRUGBANK%DB00873	Loteprednol	NR3C1	
XANTHINOL%DRUGBANK%DB09092	Xanthinol	MDH2	NNT	OGDH	GAPDH	IDH3A	RPL3	
REBOXETINE%DRUGBANK%DB00234	Reboxetine	SLC6A2	
TRIMETHADIONE%DRUGBANK%DB00347	Trimethadione	CACNA1G	
CHOLESTEROL%DRUGBANK%DB04540	Cholesterol	VDR	PCYT1B	RORA	CLEC4E	NR1I3	
ROFECOXIB%DRUGBANK%DB00533	Rofecoxib	PTGS2	ELN	
CHLOROBUTANOL%DRUGBANK%DB11386	Chlorobutanol	KCNH2	
HEXESTROL%DRUGBANK%DB07931	Hexestrol	ESR1	AKR1C1	NR1I3	ESR2	NR1I2	
MIVACURIUM%DRUGBANK%DB01226	Mivacurium	BCHE	CHRM3	CHRNA2	CHRM2	
TOLAZOLINE%DRUGBANK%DB00797	Tolazoline	DRD2	HRH2	ADRA1A	ADRA2C	ADRA2B	HRH1	ADRA2A	
TYROTHRICIN%DRUGBANK%DB13503	Tyrothricin	ACHE	
AMINOGLUTETHIMIDE%DRUGBANK%DB00357	Aminoglutethimide	CYP19A1	CYP11A1	
FERROUS ASCORBATE%DRUGBANK%DB14490	Ferrous ascorbate	TF	EGLN1	FEN1	HBA2	HDAC8	CP	POLB	NEIL2	FTH1	AHSP	NEIL1	FXN	TFRC	
CHLORPROPAMIDE%DRUGBANK%DB00672	Chlorpropamide	ABCC8	KCNJ10	
DIPHEMANIL%DRUGBANK%DB13720	Diphemanil	CHRM1	CHRM3	
CHLORTETRACYCLINE%DRUGBANK%DB09093	Chlortetracycline	ARF1	PADI4	EPHB1	PNLIP	
INDOPROFEN%DRUGBANK%DB08951	Indoprofen	PTGS2	PTGS1	CXCR1	FABP1	PKM	CXCR2	
RIMEXOLONE%DRUGBANK%DB00896	Rimexolone	NR3C1	ESRRA	
METHYCLOTHIAZIDE%DRUGBANK%DB00232	Methyclothiazide	CA2	CA1	SLC12A1	CA4	
HEXYLCAINE%DRUGBANK%DB00473	Hexylcaine	SCN10A	SCN5A	
MAGNESIUM CATION%DRUGBANK%DB01378	Magnesium cation	ATP1A1	
ASTEMIZOLE%DRUGBANK%DB00637	Astemizole	MAPT	KCNH1	HRH1	KCNH2	
CINOXACIN%DRUGBANK%DB00827	Cinoxacin	TOP2B	TOP2A	
CHLOROTRIANISENE%DRUGBANK%DB00269	Chlorotrianisene	ESR1	
LORCASERIN%DRUGBANK%DB04871	Lorcaserin	HTR2C	
DROXICAM%DRUGBANK%DB09215	Droxicam	PTGS2	PTGS1	
FINAFLOXACIN%DRUGBANK%DB09047	Finafloxacin	TOP2A	
ERYTHRITYL TETRANITRATE%DRUGBANK%DB01613	Erythrityl tetranitrate	NPR1	NPR2	
XIMELAGATRAN%DRUGBANK%DB04898	Ximelagatran	F2	
POTASSIUM CHLORIDE%DRUGBANK%DB00761	Potassium chloride	SLC12A2	SLC12A4	SLC12A5	SLC12A6	SLC12A7	SLC12A1	
PENTOXYVERINE%DRUGBANK%DB11186	Pentoxyverine	OPRK1	OPRM1	SIGMAR1	KCNH2	SCN1A	
METHOXAMINE%DRUGBANK%DB00723	Methoxamine	ADRA1D	ADRA1A	ADRA1B	
ETHCHLORVYNOL%DRUGBANK%DB00189	Ethchlorvynol	GABRA1	GABRB2	
ESTRADIOL DIENANTHATE%DRUGBANK%DB13955	Estradiol dienanthate	ESRRG	MT-ATP6	NCOA2	BECN1	GPER1	HSD17B2	ESR1	ESR2	NR1I2	CHRNA4	
PENTAERYTHRITOL TETRANITRATE%DRUGBANK%DB06154	Pentaerythritol tetranitrate	HBA2	HBB	
RITODRINE%DRUGBANK%DB00867	Ritodrine	KCNMA1	KCNJ1	ADRB2	SULT1C4	ATP2C1	MYLK	ADRB1	
DRISAPERSEN%DRUGBANK%DB13688	Drisapersen	DMD	
OMEGA-3-CARBOXYLIC ACIDS%DRUGBANK%DB09568	Omega-3-carboxylic acids	ECHS1	DGAT2	ELOVL4	LPL	HADH	HSD17B10	
CYCLIZINE%DRUGBANK%DB01176	Cyclizine	SULT1E1	HRH1	
TROVAFLOXACIN%DRUGBANK%DB00685	Trovafloxacin	TOP2A	
TRYPTOPHAN%DRUGBANK%DB00150	Tryptophan	WARS1	WARS2	IDO1	
BENOXAPROFEN%DRUGBANK%DB04812	Benoxaprofen	ACAT1	
PEMIROLAST%DRUGBANK%DB00885	Pemirolast	HRH1	
FENCAMFAMIN%DRUGBANK%DB01463	Fencamfamin	DRD2	SLC6A3	
VILOXAZINE%DRUGBANK%DB09185	Viloxazine	MAOB	MAOA	CHRM3	CHRM2	CHRM1	CHRM4	HRH2	ADRB2	HRH1	ADRA1B	SLC6A2	HTR2B	HTR2C	
AJMALINE%DRUGBANK%DB01426	Ajmaline	SCN5A	
FENDILINE%DRUGBANK%DB08980	Fendiline	HTR2B	
TIDEGLUSIB%DRUGBANK%DB12129	Tideglusib	GSK3B	
SERTINDOLE%DRUGBANK%DB06144	Sertindole	HTR2A	DRD2	ADRA1D	ADRA1A	HTR6	ADRA1B	KCNH2	HTR2C	
RESERPINE%DRUGBANK%DB00206	Reserpine	BIRC5	SLC18A1	SLC18A2	
PIPOTIAZINE%DRUGBANK%DB01621	Pipotiazine	HTR2A	DRD2	HTR1A	DRD1	
BIPERIDEN%DRUGBANK%DB00810	Biperiden	CHRM1	
IODIDE%DRUGBANK%DB12754	Iodide	CA2	CA1	
ALCLOFENAC%DRUGBANK%DB13167	Alclofenac	PTGS2	
DESERPIDINE%DRUGBANK%DB01089	Deserpidine	ACE	SLC18A2	
ZUCAPSAICIN%DRUGBANK%DB09120	Zucapsaicin	TRPV1	
LEVOBUPIVACAINE%DRUGBANK%DB01002	Levobupivacaine	SCN10A	
DOXACURIUM%DRUGBANK%DB01135	Doxacurium	CHRNA2	CHRM2	
ZIMELIDINE%DRUGBANK%DB04832	Zimelidine	MAOB	MAOA	SLC6A4	
CIANIDANOL%DRUGBANK%DB14086	Cianidanol	CA14	CA2	PTGS1	CA12	CA1	CA4	CA9	CA6	
ANCROD%DRUGBANK%DB05099	Ancrod	FGA	
ANCESTIM%DRUGBANK%DB09103	Ancestim	KIT	
DROTRECOGIN ALFA%DRUGBANK%DB00055	Drotrecogin alfa	SERPINA5	F2	PROCR	F8	PROS1	F5	SERPINB6	PF4	THBD	SERPINE1	
TILUDRONIC ACID%DRUGBANK%DB01133	Tiludronic acid	ATP6V0A1	PTPRE	PTPN6	PTPN12	
TECHNETIUM TC-99M NOFETUMOMAB MERPENTAN%DRUGBANK%DB09336	Technetium Tc-99m nofetumomab merpentan	MS4A1	EPCAM	
CHLORMEZANONE%DRUGBANK%DB01178	Chlormezanone	TSPO	
IDOXURIDINE%DRUGBANK%DB00249	Idoxuridine	TK1	
ZOMEPIRAC%DRUGBANK%DB04828	Zomepirac	PTGDR2	PTGS2	PTGS1	
ESMOLOL%DRUGBANK%DB00187	Esmolol	ADRB1	
THALIDOMIDE%DRUGBANK%DB01041	Thalidomide	CRBN	TNF	ORM1	
PLANTAGO OVATA SEED%DRUGBANK%DB14585	Plantago ovata seed	CHRM5	
NIMESULIDE%DRUGBANK%DB04743	Nimesulide	PLA2G2E	TNFSF10	LTF	PTGS2	
RETEPLASE%DRUGBANK%DB00015	Reteplase	PLG	FGA	SERPINE1	
LINDANE%DRUGBANK%DB00431	Lindane	PGR	GLRA2	GABRR1	GABRB1	GLRA3	GABRB3	GLRB	ESR1	GLRA1	NR1I2	
AMOROLFINE%DRUGBANK%DB09056	Amorolfine	SCN7A	
ALPRENOLOL%DRUGBANK%DB00866	Alprenolol	ADRB2	HTR1A	ADRB3	ADRB1	
